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Catalog/Weight Management/Tirzepatide

Tirzepatide

Tirzepatide is a dual GIP (glucose-dependent insulinotropic polypeptide) and GLP-1 receptor co-agonist, representing a next-generation incretin-based research target. The single…

$386per kit · lyophilized
Qty
1
$386
≥99.0% (HPLC/MS)CoA on every orderFree shipping on kit orders
Purity99.0%
HPLC verified · MS confirmed
FormulaC₂₂₅H₃₄₈N₄₈O₆₈
Mol. Weight4813.5 g/mol
Half-Life~5 days
FormLyophilized powder
CAS2023788-19-2
CoA Included3rd-party testedFor Research Use Only

Tirzepatide is a dual GIP (glucose-dependent insulinotropic polypeptide) and GLP-1 receptor co-agonist, representing a next-generation incretin-based research target. The single 39-amino acid molecule activates both receptor pathways, producing additive to synergistic effects on glycemic control and weight reduction compared to GLP-1 mono-agonism. Research has explored its superior efficacy in energy expenditure, adipose tissue reduction, and insulin secretion models.

Research Highlights

  • Dual GIP/GLP-1 co-agonism produces superior weight reduction vs GLP-1 alone
  • Significant reduction in HbA1c, fasting plasma glucose, and post-prandial insulin
  • Activates hypothalamic satiety centers via dual receptor mechanism
  • Superior adipose tissue reduction: subcutaneous and visceral compartments

Key References

1
Tirzepatide versus semaglutide once weekly in patients with type 2 diabetesN Engl J Med · 2021